平安! 发表于 2011-11-9 19:57 * S( v' g' u* `- C) Y) ^# ]
Pazopanib (100 mg/kg/day free base equivalent)
3 o5 B; q! q, s6 a9 q) V 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。5 w9 n, s/ ?% u& S
搜索了一下,原料一大堆。7 y9 y3 y, J, ?9 i+ S# w9 h
% O d8 E- U, p对不起!100mg/kg是用于移植瘤的,我弄错了。" y8 o/ p8 [+ }
: E/ ]4 L; \* B以下是正版说明书的推荐用量。
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* ^5 g: i' {+ F--------------------- DOSAGE AND ADMINISTRATION ----------------
( O! d( e- M0 I1 R$ g* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 2 R9 u) Y/ l, C; A( K: ]
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
1 c* k9 L7 w" } ]6 {$ N---------------------DOSAGE FORMS AND STRENGTHS --------------
7 C. E# B9 |" R- p& E2 K$ N200 mg tablets. (3)
+ k# r0 ] d7 Z, z1 H! Q1 m; J-------------------------------CONTRAINDICATIONS------------------------ |